Therapeutic potential of cyanobacterial pigment protein phycoerythrin: in silico and in vitro study of BACE1 interaction and in vivo Aβ reduction

Mukesh Ghanshyam Chaubey, Stuti Nareshkumar Patel, Rajesh Prasad Rastogi, Prabhakar Lal Srivastava, Arun Kumar Singh, Datta Madamwar, Niraj Kumar Singh

Research output: Contribution to journalArticlepeer-review

Abstract

Cyanobacteria are an immense source of innovative classes of pharmacologically active compounds exhibiting various biological activities ranging from antioxidants, antibiotics, anticancer, anti-inflammatory to anti-Alzheimer's disease. In the present study, we primarily targeted the inhibition of Beta-site amyloid precursor protein cleaving enzyme-1 (BACE1) by a naturally occurring cyanobacterial protein phycoerythrin (C-PE). BACE1 cleaves amyloid-β precursor protein (APP) and leads to accumulation of neurotoxic amyloid beta (Aβ) plaques in the brain, as an attribute of Alzheimer's disease (AD). Inhibition of BACE1 was measured in terms of their association and dissociation rate constants, thermodynamics of binding using surface plasmon resonance (SPR) and isothermal titration calorimetry (ITC). The kinetic parameters for enzyme activity were also measured using synthetic decapeptide as a substrate. We further validated the potential of PE by in-vivo histopathological staining of Aβ aggregate mutant Caenorhabditis elegans CL4176 by Thioflavin-T. The present studies pave the way for the application of naturally occurring C-PE as a putative therapeutic drug for the AD.

Original languageEnglish
Pages (from-to)368-378
Number of pages11
JournalInternational journal of biological macromolecules
Volume134
Early online date3 May 2019
DOIs
Publication statusPublished - 1 Aug 2019
Externally publishedYes

Keywords

  • Amyloid Precursor Protein Secretases/chemistry
  • Amyloid beta-Peptides/chemistry
  • Animals
  • Aspartic Acid Endopeptidases/chemistry
  • Caenorhabditis elegans
  • Cyanobacteria/chemistry
  • Enzyme Activation
  • Humans
  • Immunohistochemistry
  • Kinetics
  • Molecular Conformation
  • Molecular Docking Simulation
  • Molecular Dynamics Simulation
  • Phycoerythrin/chemistry
  • Protein Binding
  • Protein Refolding
  • Recombinant Proteins
  • Structure-Activity Relationship

Fingerprint

Dive into the research topics of 'Therapeutic potential of cyanobacterial pigment protein phycoerythrin: in silico and in vitro study of BACE1 interaction and in vivo Aβ reduction'. Together they form a unique fingerprint.

Cite this