Intramolecular epoxide ring opening cyclisation reactions involving guanidines
Research output: Contribution to journal › Article › peer-review
Electronic versions
The cyclisation of N-allyl- and N-homoallylguanidines using DMDO leading to the formation of novel 5- and 6-membered guanidine heterocycles is reported. Several of the products formed displayed weak inhibition of glycosidase enzymes.
Keywords
- guanidines, epoxides, epoxidation, DMDO, iodocyclisations, galactosidase inhibition
| Original language | English |
|---|---|
| Pages (from-to) | 845-852 |
| Number of pages | 8 |
| Journal | Tetrahedron |
| Volume | 73 |
| Issue number | 7 |
| Early online date | 27 Dec 2016 |
| DOIs | |
| Publication status | Published - 16 Feb 2017 |
Research outputs (5)
- Published
Iodocyclisations reactions of Boc- and Cbz-protected N-allylguanidines
Research output: Contribution to journal › Article › peer-review
- Published
Intramolecular palladium mediated π-allyl cyclisation of bis-Cbz- and bis-Boc-protected guanidines
Research output: Contribution to journal › Article › peer-review
- Published
Iodocyclisation and rearrangement reactions of mono-protected allyl substituted guanidines.
Research output: Contribution to journal › Article › peer-review
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